平安! 发表于 2011-11-9 19:57 - W( y) D: n! L4 V9 S
Pazopanib (100 mg/kg/day free base equivalent)
* U% @- `. u+ |$ [- Y7 X4 [ 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。+ X$ C1 d% Q; A3 M) F9 |
搜索了一下,原料一大堆。" k0 J" S% a: E4 |
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对不起!100mg/kg是用于移植瘤的,我弄错了。; a- z, n8 F* B" }* i
) G3 }0 d1 ~ X7 O以下是正版说明书的推荐用量。9 `) I8 N+ R( c0 W+ M. _5 Q
) f# c2 X" `* h7 j* `( _. N+ p# C C--------------------- DOSAGE AND ADMINISTRATION ----------------
: T6 `) I) @: O" f- w8 U$ o; x* W* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
" C; h+ f, f/ H* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
% D4 g0 I2 ?9 u( b4 G, _---------------------DOSAGE FORMS AND STRENGTHS -------------- G2 f8 _- ?! r0 o6 h+ T! [% p
200 mg tablets. (3) : L, f" q/ k5 [3 p7 e& H
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